Monograph C09AA05 - Ramipril
Propably not porphyrinogenic
PNP
Rationale
No data pointing to CYP-interactions. One reference stating probable non-porphyrinogenicity.
Risk for gastrointestinal adverse events in the form of digestive disturbances, dyspepsia, diarrhoea, nausea and vomiting motivates vigilance against insufficient intake of food, especially of carbohydrate.
Chemical description
Alanine derivative which is hydrolyzed in the liver giving rise to the ACE- inhibitor ramiprilate. Also other metabolites are produced. No data pointing to CYP-interactions. South African list: use with care.
Therapeutic characteristics
Common side effects that can be potentially porphyrinogenic through reduction in carbohydrate intake and that also can be confused with an acute porphyria attack are abdominal pain, dyspepsia, diarrhoea, nausea and vomiting. Other common side effects are muscle spasms, myalgia, headache and fatigue.
IPNet drug reports
Uneventful use reported in 29 patients with acute porphyria.
Similar drugs
Tradenames
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Ramipril Accord 1,25 mg, capsule hard · Ramipril Accord 10 mg, capsule hard · Ramipril Accord 2,5 mg, capsule hard · Ramipril Accord 5 mg, capsule hard · Ramipril Aurobindo 1,25 mg capsules, hard · Ramipril Aurobindo 1,25 mg, tabletten · Ramipril Aurobindo 10 mg, tabletten · Ramipril Aurobindo 2,5 mg capsules, hard · Ramipril Aurobindo 2,5 mg, tabletten · Ramipril Aurobindo 5 mg, tabletten · Ramipril Brillpharma 1,25 mg capsules, hard · Ramipril Brillpharma 10 mg capsules, hard · Ramipril Brillpharma 2,5 mg capsules, hard · Ramipril Brillpharma 5 mg capsules, hard · Ramipril Krka 1,25 mg, tabletten · Ramipril Krka 10 mg, tabletten · Ramipril Krka 2,5 mg, tabletten · Ramipril Krka 5 mg, tabletten · Ramipril Mylan 1,25 mg, tabletten · Ramipril Mylan 10 mg, tabletten · Ramipril Mylan 2,5 mg, tabletten · Ramipril Mylan 5 mg, tabletten · Ramipril Sandoz 1,25, tabletten 1,25 mg · Ramipril Sandoz 10, tabletten 10 mg · Ramipril Sandoz 2,5, tabletten 2,5 mg · Ramipril Sandoz 5, tabletten 5 mg Ramipril AB 10 mg comp. · Ramipril AB 2.5 mg comp. · Ramipril AB 5 mg comp. · Ramipril EG 10 mg (Impexeco) comp. · Ramipril EG 10 mg (Orifarm) comp. · Ramipril EG 10 mg comp. · Ramipril EG 2.5 mg comp. · Ramipril EG 5 mg (Impexeco) comp. · Ramipril EG 5 mg (Orifarm) comp. · Ramipril EG 5 mg comp. · Ramipril Krka 1.25 mg comp. · Ramipril Krka 10 mg comp. · Ramipril Krka 2.5 mg comp. · Ramipril Krka 5 mg comp. · Ramipril Sandoz 10 mg comp. · Ramipril Sandoz 2.5 mg comp. · Ramipril Sandoz 5 mg comp. · Tritace 10 mg (Exim Pharma) comp. · Tritace 10 mg (Orifarm) comp. · Tritace 10 mg (PI Pharma) comp. · Tritace 10 mg comp. · Tritace 2.5 mg comp. · Tritace 5 mg (Exim Pharma) comp. · Tritace 5 mg (PI Pharma) comp. · Tritace 5 mg comp. ACOVIL 10 mg COMPRIMIDOS · ACOVIL 2,5 mg COMPRIMIDOS · ACOVIL 5 mg COMPRIMIDOS · Ramipril · Ramipril Alter 10 mg Comprimidos efg · Ramipril Alter 5 mg Comprimidos efg · Ramipril Alter gen?Ricos 1,25 mg Comprimidos efg · Ramipril Alter gen?Ricos 10 mg Comprimidos efg · Ramipril Alter gen?Ricos 2,5 mg Comprimidos efg · Ramipril Alter gen?Ricos 5 mg Comprimidos efg · RAMIPRIL ARISTO 2.5 mg COMPRIMIDOS EFG · RAMIPRIL ARISTO 5 mg COMPRIMIDOS EFG · Ramipril Aristogen 10 mg Comprimidos efg · Ramipril Aristogen 5 mg Comprimidos efg · RAMIPRIL AUROBINDO 10 mg COMPRIMIDOS EFG · RAMIPRIL AUROBINDO 5 mg COMPRIMIDOS EFG · Ramipril Aurovitas 10 mg Comprimidos efg · Ramipril Aurovitas 5 mg Comprimidos efg · RAMIPRIL AUROVITAS SPAIN 2.5 mg COMPRIMIDOS EFG · RAMIPRIL BEXAL 5 mg COMPRIMIDOS EFG · RAMIPRIL CINFA 10 mg COMPRIMIDOS EFG · Ramipril Cinfa 2,5 mg Comprimidos efg · RAMIPRIL CINFA 5 mg COMPRIMIDOS EFG · RAMIPRIL COMBIX 10 mg COMPRIMIDOS EFG · RAMIPRIL COMBIX 2.5 mg COMPRIMIDOS EFG · RAMIPRIL COMBIX 5 mg COMPRIMIDOS EFG · Ramipril Krka 5 mg Comprimidos efg · RAMIPRIL NORMON 10 mg COMPRIMIDOS EFG · RAMIPRIL NORMON 2,5 mg COMPRIMIDOS EFG · RAMIPRIL NORMON 5 mg COMPRIMIDOS EFG · RAMIPRIL RATIOPHARM 10 mg COMPRIMIDOS · RAMIPRIL RATIOPHARM 2,5 mg COMPRIMIDOS · RAMIPRIL RATIOPHARM 5 mg COMPRIMIDOS · RAMIPRIL SANDOZ 10 mg COMPRIMIDOS EFG · RAMIPRIL SANDOZ 2,5 mg COMPRIMIDOS EFG · RAMIPRIL SANDOZ 5 mg COMPRIMIDOS EFG · Ramipril Stada 10 mg Comprimidos efg · Ramipril Stada 5 mg Comprimidos efg · RAMIPRIL TARBIS 2,5 mg COMPRIMIDOS EFG · RAMIPRIL TARBIS 5 mg COMPRIMIDOS EFG · RAMIPRIL TECNIGEN 10 mg COMPRIMIDOS EFG · RAMIPRIL TECNIGEN 2.5 mg COMPRIMIDOS EFG · RAMIPRIL TECNIGEN 5 mg COMPRIMIDOS EFG · Ramipril Tevagen 10 mg Comprimidos efg · Ramipril Tevagen 5 mg Comprimidos efg Eclipse · Herzatec · Krupil · Norapril · Quark · Ramipril · Tensiram · Triatec · Unipril AMPRIL 1,25 mg · AMPRIL 10 mg · AMPRIL 2,5 mg · AMPRIL 5 mg · RAMIPRIL ATB 10 mg · RAMIPRIL ATB 2,5 mg · RAMIPRIL ATB 5 mg · RAMIPRIL-AC 10 mg · RAMIPRIL-AC 2,5 mg · RAMIPRIL-AC 5 mg · TRITACE 10 mg · TRITACE 2,5 mg · TRITACE 5 mg · VIVACE 10 mg · VIVACE 2,5 mg · VIVACE 5 mg · ZENRA 10 mg · ZENRA 2,5 mg · ZENRA 5 mg Lopace · Ramipril · Ranace · Tritace Alarimed · Polpril · Ramiliv · Ramipril Aurobindo · Ramipril HEXAL · Ramipril Krka · Ramipril Stada · Ramipril Teva Ramipril Actavis · Ramipril Hexal · Triatec Ampril 10 mg tabletki · Ampril 2,5 mg tabletki · Ampril 5 mg tabletki · Apoauronarami · ApoRami · Axtil · Ivipril · Pirmamil · Polpril · Ramicor · Ramipril Actavis · Ramipril Aurobindo · Ramipril Genoptim · Ramipril Krka · Ramistad · Ramve · Tritace 10 · Tritace 2,5 · Tritace 5 · Vivace 10 mg · Vivace 2,5 mg · Vivace 5 mg Ramipril eg · Tritace Ram?l · Ramíl Cardace · Ramipril Hexal · Ramipril Orion · Ramipril Ratiopharm Cardace · Ramicor · Ramimed · Ramipril Actavis · Ramipril TAD Ampril® · Corace® · Prilinda® · Tritace® · Vivace®