Monograph A07DA03 - Loperamide
Propably not porphyrinogenic
PNP
Rationale
Synthetic opiate, some systemic absorption takes place. Probably CYP-metabolised. No data pointing to CYP-induction. Two references state non-porphyrinogenicity.
Chemical description
Synthetic opiate used in diarrhoea. Metabolized by oxidative N-demethylation. No data given on CYP-interaction, South African list: use. French list: authorized
IPNet drug reports
Uneventful use reported in 17 patients with acute porphyria.
Similar drugs
Tradenames
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Albert Heijn Diarreeremmer Loperamide HCl 2 mg, capsules · DA Diarreeremmende capsules Loperamide HCl 2 mg, harde capsules · Diarreeremmer HTP loperamide HCl 2 mg, capsules · Diarreeremmer Loperamide HCl SAM 2 mg, capsules · Etos Diarreeremmer Loperamide HCI 2 mg, capsules · Imodium 2 mg harde capsules · Imodium Instant smelttablet 2 mg orodispergeerbare tabletten · Jumbo Loperamide HCl diarreeremmer 2 mg, harde capsules · Kruidvat diarreeremmer loperamide HCl 2 mg smelttablet, orodispergeerbare tabletten · Kruidvat Loperamide HCl diarreeremmer 2 mg, harde capsules · Leidapharm Loperamide HCL diarreeremmer 2 mg, harde capsules · Livsane Diarreeremmer Loperamide HCl 2 mg, capsules · Loperamide · Loperamide HCl CF 2 mg, capsules · Loperamide HCl diarreeremmer Sameko 2 mg, harde capsules · Loperamide HCl Grindeks 2 mg harde capsules · Loperamide HCl Healthypharm 2 mg, capsules · Loperamide HCl HTP 2 mg, capsules · Loperamide HCl Linn 2 mg diarreeremmende capsules · Loperamide HCl Mylan 2 mg, capsules · Loperamide HCl RXT 2 mg diarreeremmende capsules, capsules · Loperamide HCl Sandoz 2 mg, capsules · Loperamide HCl Sanias 2 mg, harde capsules · Loperamide HCl Tenshi 2 mg, lyophilisaat voor oraal gebruik · Loperamide HCl Teva 2 mg, capsules · Loperamide HCl Triangle Pharma 2 mg diarreeremmende capsules, capsules · Loperamide HCl Viatris 2 mg, lyophilisaat voor oraal gebruik · RXT loperamide HCl 2 mg diarreeremmende capsules, capsules · Trekpleister Loperamide HCl diarreeremmer 2 mg, harde capsules Imodium · Imodium 2 mg g?l. · Imodium Instant 2 mg compr. orodisp. · Loperamide · Loperamide AB 2 mg compr. orodisp. · Loperamide AB 2 mg g?l. · Loperamide EG 2 mg g?l. · Loperamide EG Instant 2 mg compr. orodisp. · Loperamide Grindeks 2 mg g?l. · Loperamide Teva 2 mg g?l. Abeclin 2 mg Comprimidos efg · DIARFIN 2 mg CAPSULAS DURAS · Diarfin Flas 2 mg Liofilizado Oral · ELISSAN 2 mg COMPRIMIDOS · Fortasec 2 mg Capsulas Duras · FORTASEC FLAS 2 mg LIOFILIZADO ORAL · Loperamida · Loperamida Aurovitas 2 mg Capsulas Duras · Loperamida Grindeks 2 mg c?Psulas Duras · Loperamida Opko 2 mg Capsulas Duras efg · LOPERAN 2 mg CAPSULAS DURAS · Lopestop 2 mg Capsulas Duras · SALVACOLINA 0,2 mg/ml SOLUCION ORAL · SALVACOLINA 2 mg COMPRIMIDOS · Salvacolina Flas 2 mg Comprimidos Bucodispersables · SINDIAR 2 mg CAPSULAS DURAS CLORHIDRAT DE LOPERAMIDA VIM SPECTRUM 2 mg · ENTERIUM 2 mg · IMODIUM 2 mg · LOPEDIUM 2 mg · LOPEMIDOL 1 mg/5 ml · LOPEMIDOL 2 mg · LOPERAMID BIOEEL 2 mg · LOPERAMID LAROPHARM 2 mg · LOPERAMID LPH 2 mg · LOPERAMID SLAVIA 2 mg · LOPERAMID TERAPIA 2 mg · LOPERAMIDA GRINDEKS 2 mg · LOPERAMIDA LAROPHARM 1 mg/5 ml · LOPREX 2 mg · LOPRID 2 mg · TAMMEX AKUT 2 mg . · Arret · Bell's · Diah-Limit · Diaquitte · Diareze Diarrhoea Relief · Diarrhoea Relief · Diasorb · Diocalm · Diocalm Ultra · Diocaps · Dioraleze · Galpharm Diarrhoea Relief · Galpharm Loperamide · Imodium · Imodium Classic · Imodium Original · Lloydspharmacy DiaFix · Loperamide · Loritax · Norimode · Normaloe · Superdrug Loperamide Imodium · Imodium Smelt · Imolope · Lopacut · Loperamid Mashal · Loperamid Tenshi Kaizen · Soluzem Imodium · Imodium N · Imolope · Imolopera · Loperamid Norfri · Loperamid Viatris · Salvacolina AuroBlock Fast · Aurostop · Dissenten · Imodium Instant · Laremid · Lopacut · Loper · Loperamid APTEO MED · Loperamid Dr. Max · Loperamid WZF · Loperamide Aurovitas · Loperamide Grindeks · Stoperan · Stoperan FAST · Stoperan Junior · Stoperan S Imodium · Imodium Instant · Loperamid · Loperamide eg · Loperamide EG Instant Immex · Imodium · Loperamide Medical Valley Imocur · Imodium · Lopacut · Loperamide Grindeks · Loperamide Tenshi · Lopex Imodium · Imodium Instant · Lopacut · Loperamide Stirol · Loperamide-Grindeks Imodium® Instant · Loperamid Actavis · Lordiar